Conformationally Constrained Analogues of Diacylglycerol (DAG). 16. How Much Structural Complexity Is Necessary for Recognition and High Binding Affinity to Protein Kinase C?-Reference-Cited by-同舟云学术

Conformationally Constrained Analogues of Diacylglycerol (DAG). 16. How Much Structural Complexity Is Necessary for Recognition and High Binding Affinity to Protein Kinase C?

Published:2000-02-23 Issue:5 Volume:43 Page:921-944
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Nacro Kassoum¹,Bienfait Bruno¹,Lee Jeewoo¹,Han Kee-Chung¹,Kang Ji-Hye¹,Benzaria Samira¹,Lewin Nancy E.¹,Bhattacharyya Dipak K.¹,Blumberg Peter M.¹,Marquez Victor E.¹

Affiliation:

1. Laboratories of Medicinal Chemistry and of Cellular Carcinogenesis and Tumor Promotion, Division of Basic Sciences, National Cancer Institute, National Institutes of Health, Bethesda, Maryland 20892, and Laboratory of Medicinal Chemistry, College of Pharmacy, Seoul National University, Shinlim-Dong, Kwanak-Ku, Seoul 151-742, Korea

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9904607

Reference59 articles.

1. Protein Kinase C: Structure, Function, and Regulation

2. Direct Visualization of the Translocation of the γ-Subspecies of Protein Kinase C in Living Cells Using Fusion Proteins with Green Fluorescent Protein

3. Protein Kinase C as a Molecular Machine for Decoding Calcium and Diacylglycerol Signals

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