Investigation of Subsite Preferences in Aminopeptidase A (EC 3.4.11.7) Led to the Design of the First Highly Potent and Selective Inhibitors of This Enzyme-Reference-Cited by-同舟云学术

Investigation of Subsite Preferences in Aminopeptidase A (EC 3.4.11.7) Led to the Design of the First Highly Potent and Selective Inhibitors of This Enzyme

Published:1999-11-23 Issue:25 Volume:42 Page:5197-5211
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

David Christelle¹,Bischoff Laurent¹,Meudal Hervé¹,Mothé Aurélie¹,De Mota Nadia¹,DaNascimento Sophie¹,Llorens-Cortes Catherine¹,Fournié-Zaluski Marie-Claude¹,Roques Bernard P.¹

Affiliation:

1. Département de Pharmacochimie Moléculaire et Structurale, INSERM U266 − CNRS UMR 8600, UFR des Sciences Pharmaceutiques et Biologiques, 4, avenue de l'Observatoire, 75270 Paris Cedex 06, France, and Pathologie Vasculaire et Endocrinologie Rénale, INSERM U36, Collège de France, 3, rue d'Ulm, 75005 Paris Cedex, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9903040

Reference65 articles.

1. Glutamyl aminopeptidase (aminopeptidase A), the BP-1/6C3 antigen

2. Molecular cloning of the human kidney differentiation antigen gp160: human aminopeptidase A.

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