Design, Synthesis, and Biological Evaluation of C9- and C2-Substituted Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as New A2A and A3 Adenosine Receptors Antagonists-Reference-Cited by-同舟云学术

Design, Synthesis, and Biological Evaluation of C9- and C2-Substituted Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as New A2A and A3 Adenosine Receptors Antagonists

Published:2003-02-28 Issue:7 Volume:46 Page:1229-1241
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Baraldi Pier Giovanni¹,Fruttarolo Francesca¹,Tabrizi Mojgan Aghazadeh¹,Preti Delia¹,Romagnoli Romeo¹,El-Kashef Hussein¹,Moorman Allan¹,Varani Katia¹,Gessi Stefania¹,Merighi Stefania¹,Borea Pier Andrea¹

Affiliation:

1. Dipartimento di Scienze Farmaceutiche and Dipartimento di Medicina Clinica e Sperimentale-Sezione di Farmacologia, Università di Ferrara, 44100 Ferrara, Italy, Department of Chemistry, Faculty of Science, University of Assiut, Egypt, and King Pharmaceutical, 7001 Weston Parkway Suit 300, Cary, North Carolina 27513

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm021023m

Reference29 articles.

1. Structure and function of adenosine receptors and their genes

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