Allosteric Modulators of the Adenosine A1 Receptor: Synthesis and Pharmacological Evaluation of 4-Substituted 2-Amino-3-benzoylthiophenes-Reference-Cited by-同舟云学术

Allosteric Modulators of the Adenosine A1 Receptor: Synthesis and Pharmacological Evaluation of 4-Substituted 2-Amino-3-benzoylthiophenes

Published:2009-06-10 Issue:14 Volume:52 Page:4543-4547
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Aurelio Luigi¹,Valant Celine¹²,Flynn Bernard L.¹,Sexton Patrick M.¹²,Christopoulos Arthur¹²,Scammells Peter J.¹

Affiliation:

1. Medicinal Chemistry and Drug Action, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville VIC 3052, Australia

2. Drug Discovery Biology Laboratory, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Clayton VIC 3800, Australia

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9002582

Reference20 articles.

1. IV. Benzodiazepine pharmacology of cultured mammalian CNS neurons

2. Allosteric binding sites on cell-surface receptors: novel targets for drug discovery

3. Keynote review: Allosterism in membrane receptors

4. Allosteric Enhancers for A1 Adenosine Receptor

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