Development of Highly Potent and Selective Diaminothiazole Inhibitors of Cyclin-Dependent Kinases-Reference-Cited by-同舟云学术

Development of Highly Potent and Selective Diaminothiazole Inhibitors of Cyclin-Dependent Kinases

Published:2013-05-06 Issue:10 Volume:56 Page:3768-3782
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Schonbrunn Ernst¹,Betzi Stephane¹,Alam Riazul¹,Martin Mathew P.¹,Becker Andreas¹,Han Huijong¹,Francis Rawle²,Chakrasali Ramappa²,Jakkaraj Sudhakar²,Kazi Aslamuzzaman¹,Sebti Said M.¹,Cubitt Christopher L.³,Gebhard Anthony W.⁴,Hazlehurst Lori A.⁴,Tash Joseph S.⁵,Georg Gunda I.²

Affiliation:

1. Drug Discovery Department, H. Lee Moffitt Cancer Center and Research Institute, 12902 Magnolia Drive, Tampa, Florida 33612, United States

2. Department of Medicinal Chemistry, Institute for Therapeutics Discovery and Development, University of Minnesota, 717 Delaware Street SE, Minneapolis, Minnesota 55414, United States

3. Translational Research Laboratory, H. Lee Moffitt Cancer Center and Research Institute, 12902 Magnolia Drive, Tampa, Florida 33612, United States

4. Molecular Oncology Department, H. Lee Moffitt Cancer Center and Research Institute, 12902 Magnolia Drive, Tampa, Florida 33612, United States

5. Department of Molecular and Integrative Physiology, University of Kansas Medical Center, 3901 Rainbow Boulevard, Kansas City, Kansas 66160, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm301234k

Reference54 articles.

1. Protein kinase inhibitors: contributions from structure to clinical compounds

2. Genetic Alterations of Cyclins, Cyclin-Dependent Kinases, and Cdk Inhibitors in Human Cancer

3. Principles of CDK regulation

4. Cancer Cell Cycles

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