Amphipathic Benzenes Are Designed Inhibitors of the Estrogen Receptor α/Steroid Receptor Coactivator Interaction
Author:
Affiliation:
1. Department of Chemistry, University of Illinois, Urbana, Illinois 61801
2. Department of Chemistry, Cayman Chemical Company, Ann Arbor, Michigan 48108
Publisher
American Chemical Society (ACS)
Subject
Molecular Medicine,General Medicine,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/cb800056r
Reference21 articles.
1. The Structural Basis of Estrogen Receptor/Coactivator Recognition and the Antagonism of This Interaction by Tamoxifen
2. Molecular basis of agonism and antagonism in the oestrogen receptor
3. Structural Insights into the Mode of Action of a Pure Antiestrogen
4. Advanced concepts in estrogen receptor biology and breast cancer endocrine resistance: implicated role of growth factor signaling and estrogen receptor coregulators
5. Bicyclo[2.2.2]octanes: Close structural mimics of the nuclear receptor-binding motif of steroid receptor coactivators
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