Diastereoselective Synthesis of 2,3,6-Trisubstituted Piperidines-Reference-Cited by-同舟云学术

Diastereoselective Synthesis of 2,3,6-Trisubstituted Piperidines

Published:2009-05-14 Issue:12 Volume:74 Page:4525-4536
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Humphrey John M.¹,Arnold Eric P.¹,Chappie Thomas A.¹,Feltenberger John B.¹,Nagel Arthur¹,Simon Wendy¹,Suarez-Contreras Melani¹,Tom Norma J.¹,O’Neill Brian T.¹

Affiliation:

1. Pfizer Global Research and Development, Eastern Point Road, Groton, Connecticut 06340

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/jo9003184

Reference50 articles.

1. The discovery of (2S,3S)-cis-2-(diphenylmethyl)-N-[(2-methoxyphenyl)methyl]-1-azabicyclo[2.2.2]octan-3-amine as a novel, nonpeptide substance P antagonist

2. Synthesis and structure-activity relationships of CP-122,721, a second-generation NK-1 receptor antagonist

3. Studies on the active conformation of the NK1 antagonist CGP 49823. Part 21. Fluoro-olefin analogs of tertiary amide rotamers.

4. Structural Analysis and Optimization of NK1 Receptor Antagonists through Modulation of Atropisomer Interconversion Properties

5. Synthesis of (±)-CP-99994: A highly potent substance P antagonist

Cited by 17 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Enantioselective Total Synthesis of Multifidene, a Sex Pheromone of Brown Algae;Organics;2022-07-08

2. State of the Art in Crystallization‐Induced Diastereomer Transformations;Advanced Synthesis & Catalysis;2021-06-14

3. TMSOTf mediated ‘5/6-endo-dig’ reductive hydroamination for the stereoselective synthesis of pyrrolidine and piperidine derivatives;Chemical Communications;2019

4. Additive Free Fe-Catalyzed Conversion of Nitro to Aldehyde under Continuous Flow Module;ACS Sustainable Chemistry & Engineering;2018-08-14

5. Cyclic imines – preparation and application in synthesis;Organic & Biomolecular Chemistry;2018