Novel and Potent 17β-Hydroxysteroid Dehydrogenase Type 1 Inhibitors-Reference-Cited by-同舟云学术

Novel and Potent 17β-Hydroxysteroid Dehydrogenase Type 1 Inhibitors

Published:2005-03-25 Issue:8 Volume:48 Page:2759-2762
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Lawrence Harshani R.¹,Vicker Nigel¹,Allan Gillian M.¹,Smith Andrew¹,Mahon Mary F.¹,Tutill Helena J.¹,Purohit Atul¹,Reed Michael J.¹,Potter Barry V. L.¹

Affiliation:

1. Medicinal Chemistry, Department of Pharmacy and Pharmacology and Sterix Ltd., University of Bath, Claverton Down, Bath, BA2 7AY, U.K., Endocrinology and Metabolic Medicine and Sterix Ltd., Faculty of Medicine, Imperial College London, St. Mary's Hospital, London, W2 1NY, U.K., and Department of Chemistry, University of Bath, Claverton Down, Bath, BA2 7AY, U.K.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049045r

Reference25 articles.

1. Distribution of 17β-hydroxysteroid dehydrogenase gene expression and activity in rat and human tissues

2. HORMONAL THERAPY FOR BREAST CANCER

3. Steroidal regulation of oestradiol-17β dehydrogenase activity of the human breast cancer cell line MCF-7

Cited by 55 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Secosteroid diacylhydrazines as novel effective agents against hormone-dependent breast cancer cells;The Journal of Steroid Biochemistry and Molecular Biology;2024-11

2. Synthesis and Antiproliferative Activity Evaluation of B-norcholesterol-6- amide Compounds;Medicinal Chemistry;2023-10

3. N ‐Phenyl‐1,2,3,4‐tetrahydroisoquinoline: An Alternative Scaffold for the Design of 17β‐Hydroxysteroid Dehydrogenase 1 Inhibitors;ChemMedChem;2020-11-25

4. Inhibitors of 17β-hydroxysteroid dehydrogenase type 1, 2 and 14: Structures, biological activities and future challenges;Molecular and Cellular Endocrinology;2019-06

5. Synthesis of substituted 15β-alkoxy estrone derivatives and their cofactor-dependent inhibitory effect on 17β-HSD1;Journal of Enzyme Inhibition and Medicinal Chemistry;2019-01-01