Discovery of a New Nucleoside Template for Human A3 Adenosine Receptor Ligands: d-4‘-Thioadenosine Derivatives without 4‘-Hydroxymethyl Group as Highly Potent and Selective Antagonists-Reference-Cited by-同舟云学术

Discovery of a New Nucleoside Template for Human A3 Adenosine Receptor Ligands: d-4‘-Thioadenosine Derivatives without 4‘-Hydroxymethyl Group as Highly Potent and Selective Antagonists

Published:2007-06-08 Issue:14 Volume:50 Page:3159-3162
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Jeong Lak Shin¹,Choe Seung Ah¹,Gunaga Prashantha¹,Kim Hea Ok¹,Lee Hyuk Woo¹,Lee Sang Kook¹,Tosh Dilip K.¹,Patel Amit¹,Palaniappan Krishnan K.¹,Gao Zhan-Guo¹,Jacobson Kenneth A.¹,Moon Hyung Ryong¹

Affiliation:

1. Laboratory of Medicinal Chemistry, College of Pharmacy, Ewha Womans University, Seoul 120-750, Korea, Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, Bethesda, Maryland 20892, and College of Pharmacy, Pusan National University, Busan 609-753, Korea

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm070259t

Reference22 articles.

1. Adenosine receptors as therapeutic targets

2. A3 Adenosine Receptor Activation in Melanoma Cells

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