A New Structural Motif for μ-Opioid Antagonists-Reference-Cited by-同舟云学术

A New Structural Motif for μ-Opioid Antagonists

Published:2005-04-23 Issue:10 Volume:48 Page:3644-3648
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Van den Eynde Isabelle¹,Laus Georges¹,Schiller Peter W.¹,Kosson Piotr¹,Chung Nga N.¹,Lipkowski Andrzej W.¹,Tourwé Dirk¹

Affiliation:

1. Eenheid Organische Chemie, Vrije Universiteit Brussel, 2, Pleinlaan, B-1050 Brussels, Belgium, Laboratory of Chemical Biology and Peptide Research, Clinical Research Institute of Montreal, Montreal, PQ, H2W 1R7, Canada, and Medical Research Centre, Polish Academy of Sciences, Warsaw, Poland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0491795

Reference27 articles.

1. Differential stereochemical requirements of mu vs. delta opioid receptors for ligand binding and signal transduction: development of a class of potent and highly delta-selective peptide antagonists.

2. Subtleties of Structure-Agonist Versus Antagonist Relationships of Opioid Peptides and Peptidomimetics

3. The Opioid μ Agonist/δ Antagonist DIPP-NH2[Ψ] Produces a Potent Analgesic Effect, No Physical Dependence, and Less Tolerance than Morphine in Rats

4. δ Opioidmimetic Antagonists: Prototypes for Designing a New Generation of Ultraselective Opioid Peptides

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