Design, Synthesis, SAR, and Molecular Modeling Studies of Acylthiocarbamates: A Novel Series of Potent Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors Structurally Related to Phenethylthiazolylthiourea Derivatives-Reference-Cited by-同舟云学术

Design, Synthesis, SAR, and Molecular Modeling Studies of Acylthiocarbamates: A Novel Series of Potent Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors Structurally Related to Phenethylthiazolylthiourea Derivatives

Published:2003-02-01 Issue:5 Volume:46 Page:768-781
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Ranise Angelo¹,Spallarossa Andrea¹,Schenone Silvia¹,Bruno Olga¹,Bondavalli Francesco¹,Vargiu Laura¹,Marceddu Tiziana¹,Mura Massimo¹,La Colla Paolo¹,Pani Alessandra¹

Affiliation:

1. Dipartimento di Scienze Farmaceutiche, Università di Genova, Viale Benedetto XV 3, I-16132 Genova, Italy, Cooperative Laboratory IdenixUniversity of Cagliari, Cittadella Universitaria di Monserrato, 09042 Monserrato (Cagliari), Italy, and Dipartimento di Biologia Sperimentale, Università di Cagliari, Cittadella Universitaria di Monserrato, 09042 Monserrato (Cagliari), Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0209984

Reference55 articles.

1. Declining Morbidity and Mortality among Patients with Advanced Human Immunodeficiency Virus Infection

2. Novel compounds in preclinical/early clinical development for the treatment of HIV infections

3. Antiretroviral therapy: state of the HAART

4. Transmission of antiretroviral-drug-resistant HIV-1 variants

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