Synthesis and Structure−Activity Relationships of Conformationally Constrained Histamine H3 Receptor Agonists-Reference-Cited by-同舟云学术

Synthesis and Structure−Activity Relationships of Conformationally Constrained Histamine H3 Receptor Agonists

Published:2003-11-01 Issue:25 Volume:46 Page:5445-5457
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Kitbunnadaj Ruengwit¹,Zuiderveld Obbe P.¹,De Esch Iwan J. P.¹,Vollinga Roeland C.¹,Bakker Remko¹,Lutz Martin¹,Spek Anthony L.¹,Cavoy Emile¹,Deltent Marie-France¹,Menge Wiro M. P. B.¹,Timmerman Henk¹,Leurs Rob¹

Affiliation:

1. Leiden/Amsterdam Center of Drug Research (LACDR), Division of Medicinal Chemistry, Department of Pharmacochemistry, Faculty of Chemistry, Vrije Universiteit, De Boelelaan 1083, 1081 HV Amsterdam, The Netherlands, Department of Pharmaceutical Chemistry and Pharmacognosy, Faculty of Pharmaceutical Sciences, Naresuan University, Phitsanulok, Thailand, Bijvoet Center for Biomolecular Research, Department of Crystal and Structural Chemistry, Utrecht University, Padualaan 8, 3584 CH Utrecht, The Netherlands,...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm030905y

Reference54 articles.

1. Purification of a histamine H3 receptor negatively coupled to phosphoinositide turnover in the human gastric cell line HGT1.

2. Molecular Cloning and Characterization of a New Human Histamine Receptor, HH4R

3. Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

4. Histamine H3 receptors modulate the release of [3H]-acetylcholine from slices of rat entorhinal cortex: evidence for the possible existence of H3 receptor subtypes

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