Superpotent [Dmt1]Dermorphin Tetrapeptides Containing the 4-Aminotetrahydro-2-benzazepin-3-one Scaffold with Mixed μ/δ Opioid Receptor Agonistic Properties-Reference-Cited by-同舟云学术

Superpotent [Dmt1]Dermorphin Tetrapeptides Containing the 4-Aminotetrahydro-2-benzazepin-3-one Scaffold with Mixed μ/δ Opioid Receptor Agonistic Properties

Published:2011-10-20 Issue:22 Volume:54 Page:7848-7859
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Vandormael Bart¹,Fourla Danai-Dionysia²,Gramowski-Voß Alexandra³,Kosson Piotr⁴,Weiss Dieter G.³,Schröder Olaf H.-U.⁵,Lipkowski Andrzej⁴,Georgoussi Zafiroula²,Tourwé Dirk¹

Affiliation:

1. Department of Organic Chemistry, Vrije Universiteit Brussel, Pleinlaan 2, B-1050 Brussels, Belgium

2. Cellular Signaling and Molecular Pharmacology, Institute of Biology, National Centre for Scientific Research “Demokritos”, Ag. Paraskevi 15310, Athens, Greece

3. Cell Biology and Biosystems Technology, Institute of Biological Sciences, University of Rostock, 18059 Rostock, Germany

4. Medical Research Center, Polish Academy of Sciences, 02-106 Warsaw, Poland

5. NeuroProof GmbH, 18119 Rostock, Germany

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm200894e

Reference66 articles.

1. Development of Novel Enkephalin Analogues that Have Enhanced Opioid Activities at Both μ and δ Opioid Receptors

2. Opioid ligands with mixed μ/δ opioid receptor interactions: An emerging approach to novel analgesics