Evaluation of the Dmt−Tic Pharmacophore: Conversion of a Potent δ-Opioid Receptor Antagonist into a Potent δ Agonist and Ligands with Mixed Properties-Reference-Cited by-同舟云学术

Evaluation of the Dmt−Tic Pharmacophore: Conversion of a Potent δ-Opioid Receptor Antagonist into a Potent δ Agonist and Ligands with Mixed Properties

Published:2002-01-01 Issue:3 Volume:45 Page:713-720
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Balboni Gianfranco¹,Guerrini Remo¹,Salvadori Severo¹,Bianchi Clementina¹,Rizzi Daniela¹,Bryant Sharon D.¹,Lazarus Lawrence H.¹

Affiliation:

1. Department of Toxicology, University of Cagliary, I09126 Cagliary, Italy, Department of Pharmaceutical Sciences and Biotechnology Center, University of Ferrara, I-44100 Ferrara, Italy, Institute of Pharmacology, University of Ferrara, I-44100 Ferrara, Italy, and Peptide Neurochemistry, LCBRA, National Institute of Environmental Health Sciences, Research Triangle Park, North Carolina 27707

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm010449i

Reference54 articles.

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3. Selective Opioid Dipeptides

4. Schiller, P. W.; Nguyen, T. M.D.; Weltrowska, G.; Wilkes, B. C.; Marsden, B. J.; Schmidt, R.; Lemieux, C.; Chung, N. N. InPeptides:Chemistry and Biology; Hodges, R. S., Smith, J. A., Eds.; ESCOM: The Netherlands, 1994; pp 483−486.

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