Proteasome Inhibitors with Pyrazole Scaffolds from Structure-Based Virtual Screening-Reference-Cited by-同舟云学术

Proteasome Inhibitors with Pyrazole Scaffolds from Structure-Based Virtual Screening

Published:2015-02-17 Issue:4 Volume:58 Page:2036-2041
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Miller Zachary¹,Kim Keun-Sik²,Lee Do-Min¹,Kasam Vinod¹,Baek Si Eun³,Lee Kwang Hyun³,Zhang Yan-Yan⁴,Ao Lin¹,Carmony Kimberly¹,Lee Na-Ra¹,Zhou Shou¹,Zhao Qingquan¹,Jang Yujin¹,Jeong Hyun-Young⁴,Zhan Chang-Guo¹,Lee Wooin⁵,Kim Dong-Eun³,Kim Kyung Bo¹

Affiliation:

1. Department of Pharmaceutical Sciences, College of Pharmacy, University of Kentucky, Lexington, Kentucky 40536, United States

2. Department of Biomedical Laboratory Science, Konyang University, Daejeon, 302-832, Korea

3. Department of Bioscience and Biotechnology, Konkuk University, Seoul, 143-701, Korea

4. Department of Pharmacy Practice, University of Illinois at Chicago, Chicago, Illinois 60612, United States

5. College of Pharmacy, Seoul National University, Seoul, 151-742, Republic of Korea

Funder

National Cancer Institute

National Research Foundation of Korea

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm501344n

Reference42 articles.

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4. A selective inhibitor of the immunoproteasome subunit LMP7 blocks cytokine production and attenuates progression of experimental arthritis

5. Importance of the Different Proteolytic Sites of the Proteasome and the Efficacy of Inhibitors Varies with the Protein Substrate

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