Design, Synthesis, and Evaluation of Tetrasubstituted Pyridines as Potent 5-HT2C Receptor Agonists-Reference-Cited by-同舟云学术

Design, Synthesis, and Evaluation of Tetrasubstituted Pyridines as Potent 5-HT2C Receptor Agonists

Published:2015-01-27 Issue:3 Volume:6 Page:329-333
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Rouquet Guy¹,Moore Dianna E.²,Spain Malcolm,Allwood Daniel M.¹,Battilocchio Claudio¹,Blakemore David C.,Fish Paul V.,Jenkinson Stephen³,Jessiman Alan S.,Ley Steven V.¹,McMurray Gordon,Storer R. Ian

Affiliation:

1. Chemistry Department, University of Cambridge, Lensfield Road, Cambridge, CB2 1EW, U.K.

2. Worldwide Medicinal Chemistry, Pfizer Global Research and Development, Groton Laboratories, Eastern Point Road, Groton, Connecticut 06340, United States

3. Global Safety Pharmacology, Pfizer Global Research and Development, 10646 Science Center Drive, San Diego, California 92121, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml500507v

Reference24 articles.

1. Hallucinogens

2. Cardiovascular responses produced by 5-hydroxytriptamine:a pharmacological update on the receptors/mechanisms involved and therapeutic implications

3. Drugs and Valvular Heart Disease

4. New Obesity Agents: Lorcaserin and Phentermine/Topiramate

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