Turning off Transcription of the bcl-2 Gene by Stabilizing the bcl-2 Promoter Quadruplex with Quindoline Derivatives-Reference-Cited by-同舟云学术

Turning off Transcription of the bcl-2 Gene by Stabilizing the bcl-2 Promoter Quadruplex with Quindoline Derivatives

Published:2010-05-18 Issue:11 Volume:53 Page:4390-4398
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Wang Xiao-Dong¹,Ou Tian-Miao¹,Lu Yu-Jing¹,Li Zeng¹,Xu Zheng¹,Xi Chen¹,Tan Jia-Heng¹,Huang Shi-Liang¹,An Lin-Kun¹,Li Ding¹,Gu Lian-Quan¹,Huang Zhi-Shu¹

Affiliation:

1. School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou 510006, China

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm100445e

Reference54 articles.

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3. G-quadruplex formation within the promoter of the KRAS proto-oncogene and its effect on transcription

4. Characterization of the G-quadruplexes in the duplex nuclease hypersensitive element of the PDGF-A promoter and modulation of PDGF-A promoter activity by TMPyP4

5. Structure of an Unprecedented G-Quadruplex Scaffold in the Human c-kit Promoter

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