Scaling the Druggability Landscape of Human Bromodomains, a New Class of Drug Targets
Author:
Affiliation:
1. Department of Structural and Chemical Biology, Mount Sinai School of Medicine, 1425 Madison Avenue, New York, New York 10029, United States
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm3011977
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1. Chromatin Modifications and Their Function
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5. The structural basis for the recognition of acetylated histone H4 by the bromodomain of histone acetyltransferase Gcn5p
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