Discovery of Potent, Selective, Orally Active, Nonpeptide Inhibitors of Human Mast Cell Chymase-Reference-Cited by-同舟云学术

Discovery of Potent, Selective, Orally Active, Nonpeptide Inhibitors of Human Mast Cell Chymase

Published:2007-03-16 Issue:8 Volume:50 Page:1727-1730
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Greco Michael N.¹,Hawkins Michael J.¹,Powell Eugene T.¹,Almond, Harold R.¹,de Garavilla Lawrence¹,Hall Jeffrey¹,Minor Lisa K.¹,Wang Yuanping¹,Corcoran Thomas W.¹,Di Cera Enrico¹,Cantwell Angelene M.¹,Savvides Savvas N.¹,Damiano Bruce P.¹,Maryanoff Bruce E.¹

Affiliation:

1. Research and Early Development, Johnson & Johnson Pharmaceutical Research and Development, Spring House, Pennsylvania 19477-0776, and Department of Biochemistry and Molecular Biophysics, Washington University, School of Medicine, St. Louis, Missouri 63110

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0700619

Reference28 articles.

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2. Inflammation and the allergic response

3. Leukocyte granule proteins mobilize innate host defenses and adaptive immune responses

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