β-Lactones Inhibit N-acylethanolamine Acid Amidase by S-Acylation of the Catalytic N-Terminal Cysteine-Reference-Cited by-同舟云学术

β-Lactones Inhibit N-acylethanolamine Acid Amidase by S-Acylation of the Catalytic N-Terminal Cysteine

Published:2012-04-17 Issue:5 Volume:3 Page:422-426
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Armirotti Andrea¹,Romeo Elisa¹,Ponzano Stefano¹,Mengatto Luisa¹,Dionisi Mauro¹,Karacsonyi Claudia¹,Bertozzi Fabio¹,Garau Gianpiero¹,Tarozzo Glauco¹,Reggiani Angelo¹,Bandiera Tiziano¹,Tarzia Giorgio²,Mor Marco³,Piomelli Daniele¹⁴

Affiliation:

1. Department of Drug Discovery and Development, Istituto Italiano di Tecnologia, via Morego, 30, 16163 Genova, Italy

2. Dipartimento di Scienze Biomolecolari, Università degli Studi di Urbino “Carlo Bo”, Piazza del Rinascimento 6, I-61029 Urbino, Italy

3. Pharmaceutical Department, University of Parma, 43124 Parma, Italy

4. Departments of Pharmacology, University of California, Irvine, 360 MSRII, California 92697-4625, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml300056y

Reference29 articles.

1. Isolation and Structure of a Brain Constituent That Binds to the Cannabinoid Receptor

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