Indium-Labeled Macrocyclic Conjugates of Naltrindole: High-Affinity Radioligands for In Vivo Studies of Peripheral δ Opioid Receptors-Reference-Cited by-同舟云学术

Indium-Labeled Macrocyclic Conjugates of Naltrindole: High-Affinity Radioligands for In Vivo Studies of Peripheral δ Opioid Receptors

Published:2007-04-03 Issue:9 Volume:50 Page:2144-2156
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Duval Romain A.¹,Allmon Rachel L.¹,Lever John R.¹

Affiliation:

1. Departments of Radiology and the Radiopharmaceutical Sciences Institute, and Medical Pharmacology and Physiology, University of MissouriColumbia, Columbia, Missouri 65212, and Research Service, Harry S. Truman Veterans Administration Medical Center, Columbia, Missouri 65201

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0700013

Reference72 articles.

1. PET and SPECT Imaging of the Opioid System: Receptors, Radioligands and Avenues for Drug Discovery and Development

2. Synthesis of N1′-([11C]methyl)naltrindole ([11C]MeNTI): A radioligand for positron emission tomographic studies of delta opioid receptors

3. In vivo binding of N1′-([11C]methyl)naltrindole to δ-opioid receptors in mouse brain

4. Imaging of ? opioid receptors in human brain by N1?- ([11C]methyl)naltrindole and PET

5. Quantification of δ-Opioid Receptors in Human Brain with N1′ -([11C]Methyl) Naltrindole and Positron Emission Tomography

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