Diaryldiamines with Dual Inhibition of the Histamine H3 Receptor and the Norepinephrine Transporter and the Efficacy of 4-(3-(Methylamino)-1-phenylpropyl)-6-(2-(pyrrolidin-1-yl)ethoxy)naphthalen-1-ol in Pain-Reference-Cited by-同舟云学术

Diaryldiamines with Dual Inhibition of the Histamine H3 Receptor and the Norepinephrine Transporter and the Efficacy of 4-(3-(Methylamino)-1-phenylpropyl)-6-(2-(pyrrolidin-1-yl)ethoxy)naphthalen-1-ol in Pain

Published:2010-10-14 Issue:21 Volume:53 Page:7869-7873
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Altenbach Robert J.¹,Black Lawrence A.¹,Strakhova Marina I.¹,Manelli Arlene M.¹,Carr Tracy L.¹,Marsh Kennan C.¹,Wetter Jill M.¹,Wensink Erica J.¹,Hsieh Gin C.¹,Honore Prisca¹,Garrison Tiffany Runyan¹,Brioni Jorge D.¹,Cowart Marlon D.¹

Affiliation:

1. Neuroscience Research, Global Pharmaceutical Research and Development, Abbott Laboratories, 100 Abbott Park Road, Abbott Park, Illinois 60064-6100, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm100666w

Reference35 articles.

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5. The histamine H3 receptor as a therapeutic drug target for CNS disorders

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