The histamine H3 receptor: from gene cloning to H3 receptor drugs
Author:
Publisher
Springer Science and Business Media LLC
Subject
Drug Discovery,Pharmacology,General Medicine
Link
http://www.nature.com/articles/nrd1631.pdf
Reference151 articles.
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3. Arrang, J. M., Garbarg, M. & Schwartz, J. C. Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor. Nature 302, 832–837 (1983). The first description of the histamine H 3 receptor in rat brain on the basis of pharmacological data.
4. Haas, H. & Panula, P. The role of histamine and the tuberomamillary nucleus in the nervous system. Nature Rev. Neurosci. 4, 121–130 (2003). Timely review on the role of histamine in the brain.
5. Lovenberg, T. W. et al. Cloning and functional expression of the human histamine H3 receptor. Mol. Pharmacol. 55, 1101–1107 (1999). First identification of the H 3 receptor as a G-protein coupled receptor.
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