New, Non-Adenosine, High-Potency Agonists for the Human Adenosine A2B Receptor with an Improved Selectivity Profile Compared to the Reference Agonist N-Ethylcarboxamidoadenosine-Reference-Cited by-同舟云学术

New, Non-Adenosine, High-Potency Agonists for the Human Adenosine A2B Receptor with an Improved Selectivity Profile Compared to the Reference Agonist N-Ethylcarboxamidoadenosine

Published:2004-06-15 Issue:15 Volume:47 Page:3707-3709
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Beukers Margot W.¹,Chang Lisa C. W.¹,von Frijtag Drabbe Künzel Jacobien K.¹,Mulder-Krieger Thea¹,Spanjersberg Ronald F.¹,Brussee Johannes¹,IJzerman Ad P.¹

Affiliation:

1. Division of Medicinal Chemistry, LACDR, Gorlaeus Laboratories, P.O. Box 9502, 2300 RA, Leiden, The Netherlands

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049947s

Reference16 articles.

1. A Functional Screening of Adenosine Analogues at the Adenosine A2BReceptor: A Search for Potent Agonists

2. Medicinal Chemistry and Pharmacology of A2B Adenosine Receptors

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