Hydrolytic Stability versus Ring Size in Lactams: Implications for the Development of Lactam Antibiotics and Other Serine Protease Inhibitors
Author:
Affiliation:
1. Institut für Pharmazeutische Chemie, Philipps-Universität, Marbacher Weg 6, 35032 Marburg, Germany
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm000921k
Reference24 articles.
1. The β-lactamase cycle: a tale of selective pressure and bacterial ingenuity
2. [3.3.0] Pyrazolodinones: An efficient synthesis of a new class of synthetic antibacterial agents.
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