Practical Application of Oxidation Using a Novel Na2WO4−H2O2 System under Neutral Conditions for Scale-Up Manufacturing of 12α-Hydroxy-3-oxooleanano-28,13-lactone: Key Intermediate of Endothelin A Receptor Antagonist S-0139-Reference-Cited by-同舟云学术

Practical Application of Oxidation Using a Novel Na2WO4−H2O2 System under Neutral Conditions for Scale-Up Manufacturing of 12α-Hydroxy-3-oxooleanano-28,13-lactone: Key Intermediate of Endothelin A Receptor Antagonist S-0139

Published:2009-12-08 Issue:1 Volume:14 Page:289-294
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Hida Takemasa¹,Fukui Yuuki¹,Kawata Kyozo¹,Kabaki Mikio¹,Masui Toshiaki¹,Fumoto Masataka¹,Nogusa Hideo¹

Affiliation:

1. CMC Research Laboratories, Shanghai Office, Shionogi & Co., Ltd., 306A, 3F, Building A, Far East International Plaza, No. 319, Xianxia Road, Shanghai 200051, China, CMC Research Laboratories, Shionogi & Co., Ltd., 1-3, Kuise Terajima 2-chome, Amagasaki, Hyogo 660-0813, Japan, Nichia Pharmaceutical Industry, 224-20, Kawauchi Cho Hiraishi Ebisuno, Tokushima 771-0132, Japan, and Shionogi Discovery Research Laboratories, Shionogi & Co., Ltd., 12-4, Sagisu 5-chome, Fukushima-ku, Osaka 553-0002, Japan

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op900265h

Reference20 articles.

1. 13. Researches on acetylenic compounds. Part I. The preparation of acetylenic ketones by oxidation of acetylenic carbinols and glycols

2. Dimethyl sulfoxide-trifluoroacetic anhydride. New reagent for oxidation of alcohols to carbonyls

3. Readily accessible 12-I-5 oxidant for the conversion of primary and secondary alcohols to aldehydes and ketones

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