Diastereoselective Synthesis of Aryloxy Phosphoramidate Prodrugs of 3′-Deoxy-2′,3′-didehydrothymidine Monophosphate-Reference-Cited by-同舟云学术

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Diastereoselective Synthesis of Aryloxy Phosphoramidate Prodrugs of 3′-Deoxy-2′,3′-didehydrothymidine Monophosphate

Published:2010-10-14 Issue:21 Volume:53 Page:7675-7681
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Roman Cristina Arbelo¹,Balzarini Jan²,Meier Chris¹

Affiliation:

1. Organic Chemistry, Department of Chemistry, Faculty of Science, University of Hamburg, Martin-Luther-King-Platz 6, 20146 Hamburg, Germany

2. Rega Institute for Medical Research, Katholieke Universiteit Leuven, Minderbroedersstraat 10, B-3000 Leuven, Belgium

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm100817f

Reference26 articles.

1. 1,3,2-Oxathiaphospholane approach to the synthesis of P-chiral stereodefined analogs of oligonucleotides and biologically relevant nucleoside polyphosphates

2. Stereocontrolled synthesis of oligonucleoside phosphorothioates and PO/PS-chimeric oligonucleotides by using oxazaphospholidine derivatives

3. Stereocontrolled synthesis of backbone-modified oligonucleotides via diastereopure H-phosphonate intermediates

4. Intracellular delivery of bioactive AZT nucleotides by aryl phosphate derivatives of AZT

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1. Chiral Organophosphorus Pharmaceuticals: Properties and Application;Symmetry;2023-08-07

2. Prodrugs of Nucleoside 5'-Monophosphate Analogues: Overview of the Recent Literature Concerning their Synthesis and Applications;Current Medicinal Chemistry;2023-04

3. Single Diastereomers of the Clinical Anticancer ProTide Agents NUC-1031 and NUC-3373 Preferentially Target Cancer Stem Cells In Vitro;Journal of Medicinal Chemistry;2021-06-04

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5. Synthesis of Rovafovir Etalafenamide (Part III): Evolution of the Synthetic Process to the Phosphonamidate Fragment;Organic Process Research & Development;2021-05-05

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