(3-Phenylsulfonylcycloalkano[e and d]pyrazolo[1,5-a]pyrimidin-2-yl)amines: Potent and Selective Antagonists of the Serotonin 5-HT6 Receptor-Reference-Cited by-同舟云学术

(3-Phenylsulfonylcycloalkano[e and d]pyrazolo[1,5-a]pyrimidin-2-yl)amines: Potent and Selective Antagonists of the Serotonin 5-HT6 Receptor

Published:2010-06-18 Issue:14 Volume:53 Page:5186-5196
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Ivachtchenko Alexandre V.¹²,Dmitriev Dmitri E.¹,Golovina Elena S.³,Kadieva Madina G.¹,Koryakova Angela G.³,Kysil Volodymyr M.²,Mitkin Oleg D.¹,Okun Ilya M.²,Tkachenko Sergey E.²,Vorobiev Anton A.¹

Affiliation:

1. Department of Organic Chemistry

2. ChemDiv, Inc., 6605 Nancy Ridge Drive, San Diego, California 92121

3. Department of Molecular Pharmacology

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm100350r

Reference40 articles.

1. Cloning, Characterization, and Chromosomal Localization of a Human 5-HT6 Serotonin Receptor

2. The anxiolytic-like effect of the selective 5-HT6 receptor antagonist SB-399885: The impact of benzodiazepine receptors

3. Effects of the brain-penetrant and selective 5-HT6 receptor antagonist SB-399885 in animal models of anxiety and depression

4. SB-399885 is a potent, selective 5-HT6 receptor antagonist with cognitive enhancing properties in aged rat water maze and novel object recognition models

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