Evaluation and Comparison of 3D-QSAR CoMSIA Models for CDK1, CDK5, and GSK-3 Inhibition by Paullones-Reference-Cited by-同舟云学术

Evaluation and Comparison of 3D-QSAR CoMSIA Models for CDK1, CDK5, and GSK-3 Inhibition by Paullones

Published:2003-12-09 Issue:1 Volume:47 Page:22-36
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Kunick Conrad¹,Lauenroth Kathrin¹,Wieking Karen¹,Xie Xu¹,Schultz Christiane¹,Gussio Rick¹,Zaharevitz Daniel¹,Leost Maryse¹,Meijer Laurent¹,Weber Alexander¹,Jørgensen Flemming S.¹,Lemcke Thomas¹

Affiliation:

1. Institut für Pharmazie, Abteilung für Pharmazeutische Chemie, Universität Hamburg, Bundesstrasse 45, D-20146 Hamburg, Germany, Developmental Therapeutics Program, Division of Cancer Treatment and Diagnosis, National Cancer Institute, Rockville, Maryland 20852, Centre National de la Recherche Scientifique, Station Biologique, BP 74, F-29682 Roscoff, France, Department of Pharmaceutical Chemistry, University of Marburg, Marbacher Weg 6, D-35032 Marburg, Germany, and Department of Medicinal Chemistry,...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0308904

Reference58 articles.

1. GSK-3: tricks of the trade for a multi-tasking kinase

2. GSK3 takes centre stage more than 20 years after its discovery

3. Glycogen synthase kinase 3 (GSK-3) inhibitors as new promising drugs for diabetes, neurodegeneration, cancer, and inflammation

4. The Croonian Lecture 1998. Identification of a protein kinase cascade of major importance in insulin signal transduction

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