SR2067 Reveals a Unique Kinetic and Structural Signature for PPARγ Partial Agonism-Reference-Cited by-同舟云学术

SR2067 Reveals a Unique Kinetic and Structural Signature for PPARγ Partial Agonism

Published:2015-12-03 Issue:1 Volume:11 Page:273-283
ISSN:1554-8929
Container-title:ACS Chemical Biology
language:en
Short-container-title:ACS Chem. Biol.

Author:

van Marrewijk Laura M.¹,Polyak Steven W.¹,Hijnen Marcel²,Kuruvilla Dana³,Chang Mi Ra³,Shin Youseung³,Kamenecka Theodore M.³,Griffin Patrick R.³,Bruning John B.¹

Affiliation:

1. School of Biological Sciences, The University of Adelaide, Adelaide, South Australia 5005, Australia

2. GE Healthcare Life Sciences ANZ, Melbourne, Victoria 3121, Australia

3. Department of Molecular Therapeutics, The Scripps Research Institute, Scripps Florida, Jupiter, Florida 33458, United States

Funder

U.S. Department of Energy

U.S. Department of Health and Human Services

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acschembio.5b00580

Reference47 articles.

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5. Thiazolidinediones and PPARγ agonists: time for a reassessment

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