Clickable Photoaffinity Ligands for Metabotropic Glutamate Receptor 5 Based on Select Acetylenic Negative Allosteric Modulators-Reference-Cited by-同舟云学术

Clickable Photoaffinity Ligands for Metabotropic Glutamate Receptor 5 Based on Select Acetylenic Negative Allosteric Modulators

Published:2016-05-04 Issue:7 Volume:11 Page:1870-1879
ISSN:1554-8929
Container-title:ACS Chemical Biology
language:en
Short-container-title:ACS Chem. Biol.

Author:

Gregory Karen J.¹,Velagaleti Ranganadh²,Thal David M.¹,Brady Ryan M.¹,Christopoulos Arthur¹,Conn P. Jeffrey³,Lapinsky David J.²

Affiliation:

1. Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, Australia

2. Division of Pharmaceutical Sciences, Mylan School of Pharmacy, Duquesne University, Pittsburgh, Pennsylvania, United States

3. Vanderbilt Center for Neuroscience Drug Discovery and Department of Pharmacology, Vanderbilt University Medical Center, Nashville, Tennessee, United States

Funder

U.S. Department of Health and Human Services

Department of Health, Australian Government

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acschembio.6b00026

Reference38 articles.

1. Pharmacology of Metabotropic Glutamate Receptor Allosteric Modulators

2. Metabotropic glutamate receptor subtype 5: molecular pharmacology, allosteric modulation and stimulus bias