Discovery of 4,4′-Dipyridylsulfide Analogs as “Switchable Electrophiles” for Covalent Inhibition
Author:
Affiliation:
1. Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, Texas 78712, United States
Funder
National Science Foundation
Robert A Welch Foundation
Publisher
American Chemical Society (ACS)
Subject
Molecular Medicine,General Medicine,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acschembio.0c00890
Reference20 articles.
1. Covalent fragment libraries in drug discovery
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5. 2-Sulfonylpyridines as Tunable, Cysteine-Reactive Electrophiles
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