Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine Derivatives as Highly Potent and Selective Human A3 Adenosine Receptor Antagonists: Influence of the Chain at the N8 Pyrazole Nitrogen-Reference-Cited by-同舟云学术

Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine Derivatives as Highly Potent and Selective Human A3 Adenosine Receptor Antagonists: Influence of the Chain at the N8 Pyrazole Nitrogen

Published:2000-11-21 Issue:25 Volume:43 Page:4768-4780
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Baraldi Pier Giovanni¹,Cacciari Barbara¹,Romagnoli Romeo¹,Spalluto Giampiero¹,Moro Stefano¹,Klotz Karl-Norbert¹,Leung Edward¹,Varani Katia¹,Gessi Stefania¹,Merighi Stefania¹,Borea Pier Andrea¹

Affiliation:

1. Dipartimento di Scienze Farmaceutiche and Dipartimento di Medicina Clinica e Sperimentale-Sezione di Farmacologia, Università degli Studi di Ferrara, Via Fossato di Mortara 17-19, I-44100 Ferrara, Italy; Dipartimento di Scienze Farmaceutiche, Università degli Studi di Trieste, Piazzale Europa 1, I-34127 Trieste, Italy; Molecular Modeling Section, Dipartimento di Scienze Farmaceutiche, Università di Padova, Via Marzolo 5, I-35131 Padova, Italy; Institut für Pharmakologie, Universität Würzburg, Versbacher...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm001047y

Reference58 articles.

1. Recent developments in selective agonists and antagonists acting at purine and pyrimidine receptors

2. Molecular cloning of a novel putative G-protein coupled receptor expressed during rat spermiogenesis

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