Development of [18F]AmBF3 Tetrazine for Radiolabeling of Peptides: Preclinical Evaluation and PET Imaging of [18F]AmBF3-PEG7-Tyr3-Octreotide in an AR42J Pancreatic Carcinoma Model-Reference-Cited by-同舟云学术

Development of [¹⁸F]AmBF₃ Tetrazine for Radiolabeling of Peptides: Preclinical Evaluation and PET Imaging of [¹⁸F]AmBF₃-PEG₇-Tyr³-Octreotide in an AR42J Pancreatic Carcinoma Model

Published:2022-06-16 Issue:7 Volume:33 Page:1393-1404
ISSN:1043-1802
Container-title:Bioconjugate Chemistry
language:en
Short-container-title:Bioconjugate Chem.

Author:

Otaru Sofia¹^ORCID,Paulus Andreas¹^ORCID,Imlimthan Surachet¹^ORCID,Kuurne Iida¹,Virtanen Helena²,Liljenbäck Heidi²³,Tolvanen Tuula²⁴,Auchynnikava Tatsiana²⁵,Roivainen Anne²³,Helariutta Kerttuli¹^ORCID,Sarparanta Mirkka¹^ORCID,Airaksinen Anu J.¹²⁵^ORCID

Affiliation:

1. Radiochemistry, Department of Chemistry, University of Helsinki, P.O. Box 55, FI-00014 Helsinki, Finland

2. Turku PET Centre, University of Turku, Kiinamyllynkatu 4-8, FI-20520 Turku, Finland

3. Turku Center for Disease Modeling, Institute of Biomedicine, University of Turku, FI-20520 Turku, Finland

4. Department of Medical Physics, Turku University Hospital, FI-20521 Turku, Finland

5. Department of Chemistry, University of Turku, FI-20014 Turku, Finland

Funder

Academy of Finland

Jane ja Aatos Erkon S??ti?

Business Finland

Suomen Kulttuurirahasto

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Pharmaceutical Science,Pharmacology,Biomedical Engineering,Bioengineering,Biotechnology

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.bioconjchem.2c00231

Reference31 articles.

1. Synthesis of Peptide Radiopharmaceuticals for the Therapy and Diagnosis of Tumor Diseases

2. Radiolabeled Peptides: Valuable Tools for the Detection and Treatment of Cancer

3. Radiolabeled Peptides and Antibodies in Medicine

4. Effect of the positron range of 18F, 68Ga and 124I on PET/CT in lung-equivalent materials

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