Synthesis of Novel Analogs of Cabergoline: Improving Cardiovascular Safety by Removing 5-HT2B Receptor Agonism-Reference-Cited by-同舟云学术

Synthesis of Novel Analogs of Cabergoline: Improving Cardiovascular Safety by Removing 5-HT2B Receptor Agonism

Published:2013-01-14 Issue:2 Volume:4 Page:254-258
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Dosa Peter I.¹,Ward Tim¹,Walters Michael A.¹,Kim Suck Won²

Affiliation:

1. Department of Medicinal Chemistry, Institute for Therapeutics Discovery and Development, College of Pharmacy, University of Minnesota, 717 Delaware Street SE, Minneapolis, Minnesota 55414, United States

2. Department of Psychiatry, University of Minnesota Medical School, 2450 Riverside Avenue, Minneapolis, Minnesota 55454, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml3003814

Reference37 articles.

1. Cabergoline in the Treatment of Hyperprolactinemia: A Study in 455 Patients

2. Efficacy and safety of high-dose cabergoline in Parkinson's disease

3. Medical Treatment in Cushing’s Syndrome: Dopamine Agonists and Cabergoline

4. Addition of a Dopamine Agonist, Cabergoline, to a Serotonin-Noradrenalin Reuptake Inhibitor, Milnacipran as a Therapeutic Option in the Treatment of Refractory Depression: Two Case Reports

5. Cabergoline, a dopamine receptor agonist, has an antidepressant-like property and enhances brain-derived neurotrophic factor signaling

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