Probing the Binding Site of Abl Tyrosine Kinase Using in Situ Click Chemistry-Reference-Cited by-同舟云学术

Probing the Binding Site of Abl Tyrosine Kinase Using in Situ Click Chemistry

Published:2013-01-18 Issue:2 Volume:4 Page:274-277
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Peruzzotti Cristina¹,Borrelli Stella¹,Ventura Micol¹,Pantano Rebecca¹,Fumagalli Gaia¹,Christodoulou Michael S.¹,Monticelli Damiano²,Luzzani Marcello³,Fallacara Anna Lucia⁴,Tintori Cristina⁴,Botta Maurizio⁴,Passarella Daniele¹

Affiliation:

1. Dipartimento di Chimica, Università degli Studi di Milano, Via Golgi 19, 20133 Milano, Italy

2. Dipartimento di Scienze Alta Tecnologia, Università degli Studi dell’Insubria, Via Valleggio 11, 22100 Como, Italy

3. LINNEA SA, Via Cantonale, 6595 Riazzino, Switzerland

4. Dipartimento Farmaco Chimico Tecnologico, Università degli Studi di Siena, Via Alcide de Gasperi 2, I-53100, Siena, Italy

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml300394w

Reference38 articles.

1. Identification of potent c-Src inhibitors strongly affecting the proliferation of human neuroblastoma cells

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3. Design and Synthesis of Thiadiazoles and Thiazoles Targeting the Bcr-Abl T315I Mutant: from Docking False Positives to ATP-Noncompetitive Inhibitors

4. Discovery and SAR of 1,3,4-thiadiazole derivatives as potent Abl tyrosine kinase inhibitors and cytodifferentiating agents

5. C6‐Unsubstituted Pyrazolo[3,4‐d]pyrimidines Are Dual Src/Abl Inhibitors Effective against Imatinib Mesylate Resistant Chronic Myeloid Leukemia Cell Lines

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