Biarylcarbamoylindolines Are Novel and Selective 5-HT2C Receptor Inverse Agonists: Identification of 5-Methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]- 5-pyridyl]carbamoyl]-6-trifluoromethylindoline (SB-243213) as a Potential Antidepressant/Anxiolytic Agent-Reference-Cited by-同舟云学术

Biarylcarbamoylindolines Are Novel and Selective 5-HT2C Receptor Inverse Agonists: Identification of 5-Methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]- 5-pyridyl]carbamoyl]-6-trifluoromethylindoline (SB-243213) as a Potential Antidepressant/Anxiolytic Agent

Published:2000-02-25 Issue:6 Volume:43 Page:1123-1134
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Bromidge Steven M.¹,Dabbs Steven¹,Davies David T.¹,Davies Susannah¹,Duckworth D. Malcolm¹,Forbes Ian T.¹,Gaster Laramie M.¹,Ham Peter¹,Jones Graham E.¹,King Frank D.¹,Mulholland Keith R.¹,Saunders Damian V.¹,Wyman Paul A.¹,Blaney Frank E.¹,Clarke Stephen E.¹,Blackburn Thomas P.¹,Holland Vicky¹,Kennett Guy A.¹,Lightowler Sean¹,Middlemiss Derek N.¹,Trail Brenda¹,Riley Graham J.¹,Wood Martyn D.¹

Affiliation:

1. SmithKline Beecham Pharmaceuticals, Discovery Research, New Frontiers Science Park, Third Avenue, Harlow, Essex CM19 5AW, U.K.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm990388c

Reference40 articles.

1. Erratum

2. Multiple actions of somatostatin in neoplastic disease

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