Discovery of (1S,2R,3R)-2,3-Dimethyl-2-phenyl-1-sulfamidocyclopropanecarboxylates: Novel and Highly Selective Aggrecanase Inhibitors-Reference-Cited by-同舟云学术

Discovery of (1S,2R,3R)-2,3-Dimethyl-2-phenyl-1-sulfamidocyclopropanecarboxylates: Novel and Highly Selective Aggrecanase Inhibitors

Published:2011-03-21 Issue:8 Volume:54 Page:2839-2863
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Shiozaki Makoto¹,Maeda Katsuya¹,Miura Tomoya¹,Kotoku Masayuki¹,Yamasaki Takayuki¹,Matsuda Isamu¹,Aoki Kenta¹,Yasue Katsutaka¹,Imai Hiroto¹,Ubukata Minoru¹,Suma Akira¹,Yokota Masahiro¹,Hotta Takahiro¹,Tanaka Masahiro¹,Hase Yasunori¹,Haas Julia²,Fryer Andrew M.²,Laird Ellen R.²,Littmann Nicole M.²,Andrews Steven W.²,Josey John A.²,Mimura Takayuki³,Shinozaki Yuichi³,Yoshiuchi Hiromi³,Inaba Takashi¹

Affiliation:

1. Chemical Research Laboratories, Central Pharmaceutical Research Institute, Japan Tobacco Inc., 1-1 Murasaki-cho, Takatsuki, Osaka 569-1125, Japan

2. Array BioPharma Inc., 3200 Walnut Street, Boulder, Colorado 80301, United States

3. Biological Pharmacological Research Laboratories, Central Pharmaceutical Research Institute, Japan Tobacco Inc., 1-1 Murasaki-cho, Takatsuki, Osaka 569-1125, Japan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm101609j

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