Exploring the Effect of Cyclization of Histamine H1 Receptor Antagonists on Ligand Binding Kinetics
Author:
Affiliation:
1. Amsterdam Institute of Molecular and Life Sciences (AIMMS), Division of Medicinal Chemistry, Faculty of Science, Vrije Universiteit Amsterdam, De Boelelaan 1108, 1081 HZ Amsterdam, The Netherlands
Funder
Innovative Medicines Initiative
China Scholarship Council
Publisher
American Chemical Society (ACS)
Subject
General Chemical Engineering,General Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acsomega.0c06358
Reference43 articles.
1. Ligand Residence Time at G-protein–Coupled Receptors—Why We Should Take Our Time To Study It
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5. Functional efficacy of adenosine A2A receptor agonists is positively correlated to their receptor residence time
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