Side Chain Cyclization Based on Serine Residues: Synthesis, Structure, and Activity of a Novel Cyclic Analogue of the Parathyroid Hormone Fragment 1−11-Reference-Cited by-同舟云学术

Side Chain Cyclization Based on Serine Residues: Synthesis, Structure, and Activity of a Novel Cyclic Analogue of the Parathyroid Hormone Fragment 1−11

Published:2010-10-28 Issue:22 Volume:53 Page:8072-8079
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Caporale Andrea¹,Sturlese Mattia¹,Gesiot Lorenzo¹,Zanta Fabrizio¹²,Wittelsberger Angela³,Cabrele Chiara²

Affiliation:

1. Dept. of Chemical Sciences, University of Padova, Institute of Biomolecular Chemistry, CNR, via Marzolo 1, 35131 Padova, Italy

2. Fakultät für Chemie und Biochemie, Ruhr-Universität Bochum, Universitätsstrasse 150, 44801, Bochum, Germany

3. Dept. of Physiology, Tufts University School of Medicine, 136 Harrison Avenue, Boston, Massachusetts 02111, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm1008264

Reference56 articles.

1. Peptidomimetics, a synthetic tool of drug discovery

2. Current Synthetic Approaches to Peptide and Peptidomimetic Cyclization

3. Backbone Cyclic Peptidomimetic Melanocortin-4 Receptor Agonist as a Novel Orally Administrated Drug Lead for Treating Obesity

4. Downsizing human, bacterial, and viral proteins to short water-stable alpha helices that maintain biological potency

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