Backbone Cyclic Peptidomimetic Melanocortin-4 Receptor Agonist as a Novel Orally Administrated Drug Lead for Treating Obesity

Author:

Hess Shmuel1,Linde Yaniv1,Ovadia Oded1,Safrai Eli1,Shalev Deborah E.1,Swed Avi1,Halbfinger Efrat1,Lapidot Tair1,Winkler Ilan1,Gabinet Yael1,Faier Avi1,Yarden Dana1,Xiang Zhimin1,Portillo Federico P.1,Haskell-Luevano Carrie1,Gilon Chaim1,Hoffman Amnon1

Affiliation:

1. Department of Pharmaceutics, School of Pharmacy, The Hebrew University of Jerusalem, Jerusalem 91120, Israel, Institute of Chemistry, and Wolfson Centre for Applied Structural Biology, Safra Campus, Givat Ram, The Hebrew University of Jerusalem, Jerusalem 91904, Israel, Bioline Rx, Jerusalem 91450, Israel, and Department of Medicinal Chemistry, University of Florida, Gainesville, Florida 32610-0485

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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