The First Potent Inhibitors for Human Glutaminyl Cyclase: Synthesis and Structure−Activity Relationship
Author:
Affiliation:
1. Departments of Medicinal Chemistry and Enzymology, Probiodrug AG, Weinbergweg 22, 06120 Halle, Germany
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm050756e
Reference30 articles.
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3. Substrate Specificity of Glutaminyl Cyclases from Plants and Animals
4. Characterization of a 41-Residue Ovine Hypothalamic Peptide That Stimulates Secretion of Corticotropin and β-Endorphin
5. Pyrrolidone carboxyl peptidase (Pcp): An enzyme that removes pyroglutamic acid (pGlu) from pGlu-peptides and pGlu-proteins
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