3-[(2-Methyl-1,3-thiazol-4-yl)ethynyl]- pyridine: A Potent and Highly Selective Metabotropic Glutamate Subtype 5 Receptor Antagonist with Anxiolytic Activity-Reference-Cited by-同舟云学术

3-[(2-Methyl-1,3-thiazol-4-yl)ethynyl]- pyridine: A Potent and Highly Selective Metabotropic Glutamate Subtype 5 Receptor Antagonist with Anxiolytic Activity

Published:2002-12-12 Issue:2 Volume:46 Page:204-206
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Cosford Nicholas D. P.¹,Tehrani Lida¹,Roppe Jeffrey¹,Schweiger Edwin¹,Smith Nicholas D.¹,Anderson Jeffrey¹,Bristow Linda¹,Brodkin Jesse¹,Jiang Xiaohui¹,McDonald Ian¹,Rao Sara¹,Washburn Mark¹,Varney Mark A.¹

Affiliation:

1. Merck Research Laboratories, MRLSDB2, 3535, General Atomics Court, San Diego, California 92121

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm025570j

Reference21 articles.

1. Glutamate receptors in the mammalian central nervous system

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