Structural Requirements for Drug Inhibition of the Liver Specific Human Organic Cation Transport Protein 1-Reference-Cited by-同舟云学术

Structural Requirements for Drug Inhibition of the Liver Specific Human Organic Cation Transport Protein 1

Published:2008-09-13 Issue:19 Volume:51 Page:5932-5942
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Ahlin Gustav¹,Karlsson Johan¹,Pedersen Jenny M.¹,Gustavsson Lena¹,Larsson Rolf¹,Matsson Pär¹,Norinder Ulf¹,Bergström Christel A. S.¹,Artursson Per¹

Affiliation:

1. Pharmaceutical Screening and Informatics, Department of Pharmacy and Cancer Pharmacology and Informatics, Department of Medical Sciences, Uppsala University, Sweden, and AstraZeneca R&D, Mölndal, Lund, and Södertälje, Sweden

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm8003152

Reference51 articles.

1. Polyspecific Organic Cation Transporters: Structure, Function, Physiological Roles, and Biopharmaceutical Implications

2. Cloning and Characterization of Two Human Polyspecific Organic Cation Transporters

3. Cloning and Functional Expression of a Human Liver Organic Cation Transporter

4. Expression profiles of 50 xenobiotic transporter genes in humans and pre-clinical species: A resource for investigations into drug disposition

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