Novel Benzodiazepine Photoaffinity Probe Stereoselectively Labels a Site Deep within the Membrane-Spanning Domain of the Cholecystokinin Receptor-Reference-Cited by-同舟云学术

Novel Benzodiazepine Photoaffinity Probe Stereoselectively Labels a Site Deep within the Membrane-Spanning Domain of the Cholecystokinin Receptor

Published:2006-01-07 Issue:3 Volume:49 Page:850-863
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Hadac Elizabeth M.¹,Dawson Eric S.¹,Darrow James W.¹,Sugg Elizabeth E.¹,Lybrand Terry P.¹,Miller Laurence J.¹

Affiliation:

1. Department of Molecular Pharmacology and Experimental Therapeutics and Cancer Center, Mayo Clinic, Scottsdale, Arizona 85259, Department of Chemistry and Center for Structural Biology, Vanderbilt University, Nashville, Tennessee 37235-1822, Glaxo-SmithKline Research Laboratories, Research Triangle Park, North Carolina, and CGI Pharmaceuticals, Inc., Branford, Connecticut 06405

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049072h

Reference44 articles.

1. Structurally similar small molecule photoaffinity CCK-A agonists and antagonists as novel tools for directly probing 7TM receptor-ligand interactions

2. Molecular Cloning and Functional Expression of the Human Gallbladder Cholecystokinin A Receptor

3. Intrinsic photoaffinity labeling probes for cholecystokinin (CCK)-gastrin family receptors. D-Tyr-Gly-[Nle28,31,pNO2-Phe33)CCK-26-33).

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