Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-Associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity-Reference-Cited by-同舟云学术

Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-Associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity

Published:2011-06-13 Issue:13 Volume:54 Page:4928-4932
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Cheng Donghang¹,Valente Sergio²,Castellano Sabrina³,Sbardella Gianluca³,Di Santo Roberto²,Costi Roberta²,Bedford Mark T.¹,Mai Antonello²

Affiliation:

1. The University of Texas MD Anderson Cancer Center, Science Park—Research Division, Smithville, Texas 78957, United States

2. Istituto Pasteur—Fondazione Cenci Bolognetti, Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza Università di Roma, P.le A. Moro 5, 00185 Roma, Italy

3. Dipartimento di Scienze Farmaceutiche e Biomediche, Università degli Studi di Salerno, Via Ponte Don Melillo, 84084 Fisciano (SA), Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm200453n

Reference28 articles.

1. Protein Arginine Methylation in Mammals: Who, What, and Why

2. Arginine Methylation

3. Chemical mechanisms of histone lysine and arginine modifications

4. Specific regional distribution of protein arginine methyltransferase 8 (PRMT8) in the mouse brain

5. Regulation of Transcription by a Protein Methyltransferase

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