Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor

Author:

Feoli Alessandra1ORCID,Iannelli Giulia12,Cipriano Alessandra1,Milite Ciro1ORCID,Shen Lei3,Wang Zhihao3,Hadjikyriacou Andrea4ORCID,Lowe Troy L.4,Safaeipour Cyrus4,Viviano Monica1ORCID,Sarno Giuliana12,Morretta Elva5,Monti Maria Chiara5ORCID,Yang Yanzhong3,Clarke Steven G.4,Cosconati Sandro6ORCID,Castellano Sabrina1ORCID,Sbardella Gianluca1ORCID

Affiliation:

1. Department of Pharmacy, Epigenetic Med Chem Lab, University of Salerno, via Giovanni Paolo II 132, Fisciano ,I-84084 SA Italy

2. PhD Program in Drug Discovery and Development, University of Salerno, via Giovanni Paolo II 132, Fisciano ,I-84084 SA Italy

3. Department of Cancer Genetics and Epigenetics, Beckman Research Institute, City of Hope National Cancer Center, Duarte, California 91010, United States

4. Department of Chemistry and Biochemistry, and the Molecular Biology Institute, University of California, Los Angeles, California 90095, United States

5. Department of Pharmacy, ProteoMass Lab, University of Salerno, via Giovanni Paolo II 132, Fisciano ,I-84084 SA Italy

6. DiSTABiF, University of Campania “Luigi Vanvitelli”, Via Vivaldi 43, 81100 Caserta, Italy

Funder

Division of Molecular and Cellular Biosciences

Ministero dell’Istruzione, dell’Università e della Ricerca

Associazione Italiana per la Ricerca sul Cancro

Università degli Studi di Salerno

National Institute of General Medical Sciences

Regione Campania

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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