An Efficient Process for the Large-Scale Synthesis of a 2,3,6-Trisubstituted Indole-Reference-Cited by-同舟云学术

An Efficient Process for the Large-Scale Synthesis of a 2,3,6-Trisubstituted Indole

Published:2012-11-26 Issue:12 Volume:16 Page:1947-1952
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Alorati Anthony D.¹,Gibb Andrew D.¹,Mullens Peter R.¹,Stewart Gavin W.¹

Affiliation:

1. Global Process Chemistry, Merck Sharp & Dohme Ltd, Hertford Road, Hoddesdon, Hertfordshire EN11 9BU, United Kingdom

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op300303p

Reference30 articles.

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2. bHudyma, T. W.; Zheng, X.; He, F.; Ding, M.; Bergstrom, C. P.; Hewawasam, P.; Martin, S. W.; Gentles, R. G.PCT Int. Appl. WO/2006/020082, 2006.

3. cConte, I.; Ercolani, C.; Narjes, F.; Pompei, M.; Rowley, M.; Stansfield, I.PCT Int. Appl. WO/2006/046030, 2006.

4. Discovery of Conformationally Constrained Tetracyclic Compounds as Potent Hepatitis C Virus NS5B RNA Polymerase Inhibitors

5. eHudyma, T. W.; Zheng, X.; He, F.; Ding, M.; Bergstrom, C. P.; Hewawasam, P.; Martin, S. W.; Gentles, R. G.PCT Int. Appl. WO/2007/092000, 2007.

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