Rational Design and Simple Chemistry Yield a Superior, Neuroprotective HDAC6 Inhibitor, Tubastatin A-Reference-Cited by-同舟云学术

Rational Design and Simple Chemistry Yield a Superior, Neuroprotective HDAC6 Inhibitor, Tubastatin A

Published:2010-07-09 Issue:31 Volume:132 Page:10842-10846
ISSN:0002-7863
Container-title:Journal of the American Chemical Society
language:en
Short-container-title:J. Am. Chem. Soc.

Author:

Butler Kyle V.¹,Kalin Jay¹,Brochier Camille¹,Vistoli Guilio¹,Langley Brett¹,Kozikowski Alan P.¹

Affiliation:

1. Drug Discovery Program, Department of Medicinal Chemistry and Pharmacognosy, University of Illinois at Chicago, 833 South Wood, Chicago, Illinois 60612, Burke Medical Research Institute, 785 Mamaroneck Avenue, White Plains, New York 10605, and Dipartimento di Scienze Farmaceutiche “Pietro Pratesi”, Università degli Studi di Milano, Via Mangiagalli 25, I-20133 Milan, Italy

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

Link

https://pubs.acs.org/doi/pdf/10.1021/ja102758v

Reference29 articles.

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4. Histone Deacetylase Inhibitors: Overview and Perspectives

5. Histone deacetylases (HDACs): characterization of the classical HDAC family

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