Anomalous Role Change of Tertiary Amino and Ester Groups as Hydrogen Acceptors in Eudragit E Based Solid Dispersion Depending on the Concentration of Naproxen-Reference-Cited by-同舟云学术

Anomalous Role Change of Tertiary Amino and Ester Groups as Hydrogen Acceptors in Eudragit E Based Solid Dispersion Depending on the Concentration of Naproxen

Published:2015-03-03 Issue:4 Volume:12 Page:1050-1061
ISSN:1543-8384
Container-title:Molecular Pharmaceutics
language:en
Short-container-title:Mol. Pharmaceutics

Author:

Ueda Hiroshi¹²,Wakabayashi Shinobu¹,Kikuchi Junko¹,Ida Yasuo¹,Kadota Kazunori²,Tozuka Yuichi²

Affiliation:

1. Physicochemical and Preformulation, Applied Chemistry for Drug Discovery, Innovative Drug Discovery Research Laboratories, Shionogi & Co., Ltd., 3-1-1, Futaba-cho, Toyonaka-shi, Osaka 561-0825, Japan

2. Laboratory of Formulation Design and Pharmaceutical Technology, Osaka University of Pharmaceutical Sciences, 4-20-1, Nasahara, Takatsuki-shi, Osaka 569-1094, Japan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Pharmaceutical Science,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/mp5005417

Reference46 articles.

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2. Polymer Combination Increased Both Physical Stability and Oral Absorption of Solid Dispersions Containing a Low Glass Transition Temperature Drug: Physicochemical Characterization and in Vivo Study

3. Pharmaceutical Applications of Solid Dispersion Systems

4. Soluplus® as an effective absorption enhancer of poorly soluble drugs in vitro and in vivo

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